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Patent Search
 
Patent Guide
 

Presentations, Invited Speaker and Patents

 

Feb 2020 - Guest Speaker (Converse College, Spartanburg SC) "Careers in Science: Science and Technology Prospects and Outlook"

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Dec 2017 - Annual Seminars & Workshops (Clemson University) "Bridging the Gap Between Industry & Academia"

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May 2014 - 13th Annual Cambridge Health Tech Institute’s Conference (World Pharma Congress) “Exploring and Optimizing Cost-Effective Route Toward DPP-IV Inhibitor Compounds”. Efficient Process Chemistry (Successes and Challenges in API Development; interview Podcast)

 

April 2011 - AACR Annual Meeting, Orlando FL

“Characterization of a Novel Class of p70S6K1 (S6K1) Inhibitors in Preclinical Models”

 

June 2010 - The 32nd National Medicinal Chemistry Symposium, Minneapolis, MN

“Identification and Characterization of Small Molecule Inhibitors of the p70S6K1 (S6K1)”

 

August 2008 - The 236th ACS National Meeting, Philadelphia, PA

“Design, Synthesis, and Biological Evaluation of Novel Pyridoazepine Derivatives as Potent and Selective Serotonin 5-HT2C Receptor Agonist”

 

March 2004 – 227th ACS National Meeting, Anaheim, CA

"Investigation of Transition Metal-mediated Supramolecular self-assemblies Featuring Endohedral Ethylenediamine Palladium (II) Moieties"

 

June 2003 – 58th Northwest Regional Meeting of the American Chemical Society, Bozeman, MT

"A Total synthesis of Antitumor Agent, (-)-Epothilone B"

 

June 2001 - 37th National Organic Symposium, Bozeman, MT

“Studies of Nucleophile Ring Opening of Oxabicyclic Systems in Highly Polar Media: Application to A Total Synthesis of Antitumor Agent, (-)-Epothilone B"

 

 

U.S. and International Issued Patents

 

  • “Synthesis of Heterocyclic Compounds” Diep, K. N.; Araldi, Gian-Luca.; Ronsheim, M.; Zhou, Shao Hong. U.S. Patent #7511150 (Mar 31, 2009).

 

  • “Substituted Imidazopyrimidines and Imidazopyridines as Cannabinoid Receptor Ligands” Diep, K. N.; Araldi, Gian-Luca.; Ronsheim, M. U.S. Patent #7563797 (July 21, 2009).

 

  • “Arylamino N Heteroaryl Compounds As Mek Inhibitors” Diep, K. N.; Goutopoulos, A.; Askew, C. B.; Karra, Srinivasa.; Schwarz, M.; Yu, Henry. U.S. Patent #7772233 (Aug 10, 2010).

 

  • Pyridoazepine Derivatives” Diep, K. N.; Araldi, Gian-Luca.; Bischoff, A. U.S. Patent #7897595 (Mar 1, 2011).

 

  • “Arylamino N Heteroaryl Compounds As Mek Inhibitors”, (Claims priority): Diep, K. N.; Goutopoulos, A.; Askew, C. B.; Karra, Srinivasa.; Schwarz, M.; Yu, Henry. U.S. Patent #8802703 (Aug 12, 2014).

 

  • “Methods for The Synthesis of 1,3-Substituted Amino Uracils and Other Xanthine-Related Compounds” Diep, K. N.; Yuriy, K. U.S. Patent #9221821 (Dec 29, 2015).

 

  • “Synthesis of Beta-Arrestin Effectors” Diep, K. N.; Yuriy, K.; Graham, L.; Ronsheim, M; Zhou, Shao Hong;        

       Racha, Saibaba. U.S. Patent #9611293 (April 4, 2017)

 

Published U.S. and International Patent Applications

 

  • “Piperidine Derivatives Useful as Melanocortin Receptor Ligands” Diep, K. N.; Araldi, Gian-Luca. U.S. Patent Application #60/867,208.

 

  •  “p-70S6K Kinase Inhibitor-Phthalazine Derivatives” Diep, K. N.; Araldi, Gian-Luca.;  Ronsheim, Melanie.; Ronsheim, Mathew. U.S. Patent Application #11/939,564.

 

  • “Imidazopyridine and Imidazopyrimidine Derivatives” Diep, K. N.; Araldi, Gian-Luca.; Ronsheim, M. U.S. Patent Application #11/845,117; WO 2008/027812.

 

  •  “Methods for Preparing Dipeptidyl Peptidase IV (DPP-IV) Inhibitor Compounds” Diep, K. N.; Yuriy, K.; Graham, L.; Ronsheim, M. U.S. Patent Application #12/724,775; WO 2010/107809.

 

  • “Novel Arylamino N-Heteraryls as MEK Inhibitors” Diep, K. N.; Goutopoulos, A.; Askew, C. B.; Karra, Srinivasa.; Schwarz, M.; Yu, Henry. U.S. Patent Application #12/815,071; WO 2007/123939.

 

  • “Beta-Arrestin Effectors” Diep, K. N.; Yuriy, K.; Graham, L.; Ronsheim, M; Zhou, Shao Hong; Racha, Saibaba. U.S. Patent Application #15796438.8-1466; WO 2015/179349; US2015031497.

 

  •  “Methods for Preparing Enzyme Dipeptidyl Peptidase IV (DPP-IV)- 2nd Generation Synthesis of Dutogliptin” Diep, K. N.; Yuriy, K.; Ronsheim, M. Provisional U.S. patent filed.

 

  • “Synthesis of Glucokinase Activator Chiral Sulfoxide, GK1-399 via Kinetic Oxidation” Diep, K. N. Provisional U.S. patent filed.

 

  •  “Enantioselective Process for Preparing Intermediates of Pleuromutilin Derivatives” Diep, K. N.; Ronsheim, M. Provisional U.S. patent filed.

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  • "Sulfoxide and Sulfone Glucokinase Activators and Methods of Use Thereof" Diep, K. N.; Ronsheim, M; Pitchen, P. Provisional U.S. patent filed.

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